Browsing UTSA Faculty and Staff Works by Author "Marichev, Kostiantyn"

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Chiral donor−acceptor azetines as powerful reactants for synthesis of amino acid derivatives

Doyle, Michael; Marichev, Kostiantyn; Dong, Kuiyong; Massey, Lynée; Deng, Yongming; De Angelis, Luca; Wang, Kan; Arman, Hadi (Nature Communications;, 2019-11-22)

Coupling reactions of amines and alcohols are of central importance for applications in chemistry and biology. These transformations typically involve the use of a reagent, activated as an electrophile, onto which nucleophile ...
Highly selective acylation of polyamines and aminoglycosides by 5-acyl-5-phenyl-1,5-dihydro-4H-pyrazol-4-ones

Doyle, Michael; Marichev, Kostiantyn; Garcia, Estevan; Bhowmick, Kartick; Wherritt, Daniel J.; Arman, Hadi (Chemical Science;, 2017-08-30)

5-Acyl-5-phenyl-1,5-dihydro-4H-pyrazol-4-ones, accessible from arylpropargyl phenyldiazoacetates, are highly selective acyl transfer reagents for di- and polyamines, as well as aminoalcohols and aminothiols. As reagents ...